| Term | Definition |
| Botulinum toxin Type A | Ach blocker |
| Methyldopa | A agonist (Hypertension) |
| Darifenacin | M3 antagonist (Overactive Bladder) |
| Phenylephrine | (Selective) A1 agonist |
| Clonidine | A2 agonist (Hypertension) |
| Dobutamine | B1 agonist (Increase Cardiac Output) |
| Terbutaline | (Selective) B2 agonist (Bronchodilation) |
| Metroprolol | B1 antagonist (Hypertension) |
| Atenolol | B1 antagonist (Hypertension) |
| Prazosin | A1 antagonist (Hypertension) |
| Imipramine | NET blocker (Depression) |
| Entacapone | COMT inhibitor (peripheral, treats Parkinson's) |
| Tolcapone | COMT inhibitor (brain) |
| Tranylcypromine | MAO antagonist (treats depression) |
| Reserpine | VAMT-2 Blocker (Hypertension) |
| Propranolol | B antagonist (non-selective) |
| Phenoxybenzamine | A antagonist (nonselective, treats hypertension) |
| Selegiline | MAO-b inhibitor (selective, treats parkinson's) |
| Phenelzine | MAO antagonist |
| Isocarboxazid | MAO antagonist |
| Bretylium | NE blocker |
| Guanedrel | NE blocker |
| Guanethidine | NE blocker |
| Trimethaphan | Ganglionic blocker |
| Hexamethonium | Ganglionic blocker |
| Succinylcholine | Depolarizing agent (ACh mimic) |
| Tubocurarine | Neuromuscular blockade (blocks transmission at motor endplates) |
| Pirenzapine | M1 agonist |
| Tripitramine | M2 agonist |
| Isoproterenol | B agonist (non-selective) |
| Moclobemide | MAO-a inhibitor (selective) |
| Pargyline | MAO inhibitor |
| Nialamide | MAO antagonist |
| Ephedrine | Sympathomimetic |
| Tyramine | Sympathomimetic |
| α-methyltyrosine | NE blocker (synthesis) |
| Cocaine | NET blocker |
| Yohimbine | A2 antagonist |
| Hemicholinium | Choline uptake blocker |
| Vesamicol | ACh inhibitor |
| Atropine | M antagonist (anticholinesterase overdose) |
| Bethanechol | M agonist (urinary tract motility) |
| Pilocarpine | M agonist (xerostomia/dry mouth) |
| Cevimeline | M agonist (xerostomia/dry mouth) |
| Scopolamine | M antagonist (motion sickness) |
| Homatropine | M antagonist (dilated pupils/eye muscle paralysis) |
| Tropicamide | M antagonist (overactive bladder) |
| Ipratropium | M antagonist (COPD/Asthma) |
| Tolterodine | M antagonist (overactive bladder) |
| Oxybutynin | M antagonist (overactive bladder) |
| Trospium | M antagonist (overactive bladder) |
| Solifenacin | (selective) M3 antagonist (overactive bladder) |
| Flavoxate | M antagonist (urinary disorders) |
| Hyoscyamine | M antagonist (irritable bowel syndrome) |
| Benztropine | M antagonist (parkinson's) |
| Trihexyphenidyl | M antagonist (parkinson's) |
| Glycopyrrolate | M antagonist (irritable bowel syndrome) |
| Methscopolamine | M antagonist (irritable bowel syndrome) |
| Tiotropium | M antagonist (COPD/Asthma) |
| Methecholine | M agonist (diagnosis of asthma) |
| Dicyclomine | M antagonist (irritable bowel syndrome) |
| Acetylcholine | M agonist (miosis during opthalmic surgery) |
| Metoclopramide | M antagonist (GI motility) |
| Propantheline | M antagonist (overactive bladder) |
| Mepenzolate | M antagonist (peptic ulcer disease) |
| Carbachol | M agonist (glaucoma) |
| Echothiophate | AChase Inhibitor (open angle glaucoma) |
| Physostigmine | AChase Inhibitor (reverses anticholinergic activity/Induce paralysis during surgery) |
| Neostigmine | AChase Inhibitor (impaired function of motor nerve impulse) |
| Edrophonium | AChase Inhibitor (short acting/diagnose impaired motor nerve impulse) |
| Donepezil | AChase Inhibitor (Alzheimers) |
| Tacrine | AChase Inhibitor (Alzheimers) |
| Rivastigmine | AChase Inhibitor (Alzheimers) |
| Pyridostigmine | Achase Inhibitor (Glaucoma/Gastrourinary motility) |
| Galantamine | AChase Inhibitor (Alzheimers) |
| Demecarium | AChase Inhibitor (open angle glaucoma) |
| Ambenonium | AChase Inhibitor (Glaucoma/Gastrourinary motility) |
| Pralidoxime | AChase Inhibitor (reactivator) |