| Term | Definition |
| 3A4 IND | St. John's Wort |
| 2C19 INH, 2D6 INH | fluoxetine |
| 1A2 INH, 2C19 INH, 3A4 INH | fluvoxamine |
| 2D6 INH | paroxetine |
| 2D6 INH | bupropion |
| 1A2 SUB, 3A4 SUB | clozapine |
| 1A2 SUB | olanzapine |
| 1A2 SUB, 2C19 SUB, 2D6 SUB, 3A4 SUB | clomipramine |
| 1A2 SUB, 2C19 SUB, 2D6 SUB, 3A4 SUB | imipramine |
| 1A2 SUB, 2C19 SUB, 2D6 SUB, 3A4 SUB | amitriptyline |
| 2C9 SUB, 2C19 SUB, 3A4 IND | phenytoin |
| 2C19 SUB | diazepam |
| 2C19 SUB | DESMETHYLDIAZEPAM |
| 2D6 SUB | all TCAs |
| 2D6 SUB | atomoxetine |
| 3A4 SUB | midazolam |
| 3A4 SUB, 3A4 IND | carbamazepine |
| 2D6 INH and SUB, 3A4 SUB | haloperidol |
| 2D6 INH | phenothiazine |
| 2C9 IND, 3A4 IND | barbiturates (generally) |
| 1A2 SUB | CAFFEINE |
| 1A2 SUB | THEOPHYLLINE |
| 1A2 SUB | R-WARFARIN |
| 2C9 SUB | S-WARFARIN |
| 2D6 SUB | METOPROLOL |
| 2D6 SUB | PROPAFENONE |
| 2D6 SUB | CODEINE |
| 2D6 SUB | DEXTROMETHORPHAN |
| 2D6 SUB | TRAMADOL |
| 3A4 SUB | Ca2+ CHANNEL BLOCKERS |
| 3A4 SUB | SIMVASTATIN |
| 3A4 SUB | ATORVOSTATIN |
| 3A4 SUB | LOVASTATIN |
| 3A4 SUB | CYCLOSPORINE |
| 3A4 SUB | TACROLIMUS |
| 3A4 SUB, 2D6 INH, 3A4 INH | RITONAVIR |
| 3A4 SUB | ESTROGENS |
| 3A4 SUB | PIMOZIDE |
| 3A4 SUB, 3A4 IND | CARBAMAZEPINE |
| 1A2 INH, 2C19 INH, 2D6 INH | CIMETIDINE |
| 1A2 INH, 2C9 INH, 2D6 INH | AMIODARONE |
| 1A2 INH, 2C9 INH, 3A4 INH | DISULFIRAM |
| 1A2 INH | CIPROFLOXACIN |
| 1A2 INH | LEVOFLOXACIN |
| 1A2 INH | ENOXACIN |
| 1A2 INH | NORFLOXACIN |
| 2C9 INH | ZAFIRLUKAST |
| 2C19 INH | LANSOPRAZOLE |
| 2C19 INH | OMEPRAZOLE |
| 2C19 INH | TOPIRAMATE |
| 2D6 INH | QUINIDINE |
| 2D6 INH | TERBINAFINE |
| 3A4 INH | DILTIAZEM |
| 3A4 INH | CLARITHROMYCIN |
| 3A4 INH | ERYTHROMYCIN |
| 3A4 INH | GRAPEFRUIT JUICE |
| 3A4 INH | QUININE |
| 3A4 INH | INDINAVIR |
| 3A4 INH | NEFAZODONE |
| 3A4 INH | NELFINAVIR |
| 3A4 INH | SAQUINAVIR |
| 3A4 INH | KETOCONAZOLE |
| 3A4 INH | ITRACONAZOLE |
| 3A4 SUB, 3A4 INH | VERAPAMIL |
| 1A2 IND | TOBACCO |
| 2C9 IND, 3A4 IND | RIFAMPIN |
| 2C9 IND, 3A4 IND | PHENOBARTIBAL |
| 2D6 SUB, 3A4 SUB | ARIPIPRAZOLE |
| 2D6 SUB | RISPERIDONE |
| 3A4 SUB | ZIPRASIDONE |
| 3A4 SUB | QUETIAPINE |
| 2D6 SUB | FLUPHENAZINE |
| 2D6 SUB | PERPHENAZINE |