Set: Pharmacology test 2

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All 106 Terms

Term Definition
Trazodone, Nefazodone Antidepressants; Inhibit reuptake of 5-HT, block post-synaptic 5-HT2 receptors (2)
Bupropion Antidepressant; Inhibits DA, 5-HT, and NE uptake
Mirtazapine Antidepressant; Alpha2 antagonist (increased NE and 5-HT), H1 receptor antagonist
Fluoxetine, Sertraline Antidepressants; SSRIs (can inhibit P-450s, anorgasmia) (2)
Venlafaxine, Duloxetine Antidepressants; SNRIs (2)
Amitriptyline, Nortriptyline, Imipramine, Desipramine Antidepressants; TCAs (4)
Tranylcypromine, Phenelzine, Isocarboxazid Antidepressants; MAOIs (nonselective)--Atypical depression (3)
Selegiline Antidepressant; MAOI (type b)
Lithium, Valproic acid, Carbamazepine, Lamotrigine Antidepressants; For bipolar patients (4)
Phenytoin, Carbamazepine, Oxcarbazepine, Phenobarbital, Gabapentin, Tiagabine, Levetiracetam, Felbamate Antiepileptics; For partial and generalized tonic-clonic seizures (8)
Ethosuximide Antiepileptic; For absence seizures
Valproic acid, Lamotrigine, Topiramate, Zonisamide Antiepileptics; For a variety of seizure types (4)
Lorazepam, Diazepam, Fosphenytoin Antiepileptics; For status epilepticus (3)
Vigabatrin, Corticotropin, Prednisone Antiepileptics; For infantile spasms (3)
Anakinra Immunomodulators; Cytokines and growth factors; Cytokine antagonists; IL-1 receptor antagonist
Terbutaline, albuterol, salmeterol Asthma; Bronchodilators; Beta-adrenergic agonists (3)
Ipratropium Asthma; Bronchodilators; Muscarinic antagonist
Theophylline, aminophylline Asthma; Bronchodilators; Methylxanthines (2)
Beclomethasone, fluticasone, budesonide, prednisone Asthma; Anti-inflammatory agents; corticosteroids (4)
Zileuton, zafirlukast, montelukast Asthma; Anti-inflammatory agents; Leukotriene pathway modifiers (3)
Cromolyn, nedocromil Asthma; Anti-inflammatory agents; release inhibitors (2)
Omalizumab Asthma; Anti-inflammatory agents; anti-IgE therapy
Dimenhydrinate, diphenhydramine, meclizine, promethazine, fexofenadine, loratadine Autocoids; Antihistamines (6)
Dramamine Autocoids; Antihistamines; Dimenhydrinate trade name
Benadryl Autocoids; Antihistamines; Diphenhydramine trade name
Antivert Autocoids; Antihistamines; Meclizine trade name
Phenergan Autocoids; Antihistamines; Promethazine trade name
Allegra Autocoids; Antihistamines; Fexofenadine trade name
Claritin Autocoids; Antihistamines; Loratadine trade name
Sumatriptan Autocoids; Biogenic Amines; Triptans; For migraine use; 5-HT1 agonist
Bismuth subsalicylate (Pepto-Bismol) GI drugs; Mucosal protective agent
Cimetidine, Ranitidine GI drugs; H2-receptor antagonists (2)
Omeprazole, esomeprazole, rabeprazole Proton pump inhibitors (3)
Misoprostol GI drugs; Prostaglandin (prostaglandin E1 analog), abortifactant
Metoclopramide GI drugs; Prokinetic agent (D2 antagonist, 5-HT3 antagonist, 5-HT4 agonist)
Metoclopramide, chlorpromazine, prochlorperazine, promethazine, droperidol GI drugs; Antiemetics; D2 receptor antagonists (5)
Odansetron, granisetron, palonsetron GI drugs; Antiemetics; 5-HT3 receptor antagonists (3)
aprepitant GI drugs; Antiemetics; Substance P antagonist
Dimenhydrinate GI drugs; Antiemetics; H1 antihistamine
Nabilone GI drugs; Antiemetics; Cannabinoid
Sulfasalazine, mesalamine GI drugs; Inflammatory bowel disease (2)
Cyclosporine, Tacrolimus, Pimecrolimus Immunomodulators; Calcineurin inhibitors (3)
Sirolimus, mycophenolate mofetil, leflunomide, thalidomide Immunomodulators; Regulators of cytokine response (4)
Azathioprine Immunomodulators; Purine analog
Methotrexate Immunomodulators; For autoimmune diseases
Glatiramer Immunomodulators; Similar to myelin basic protein; for MS
Anakinra Immunomodulators; Cytokine antagonist
Leflunomide Immunomodulators; Regulators of cytokine response; inhibits dihydroorotate dehyrogenase
Infliximab Immunomodulators; Monoclonal antibodies; monoclonal antibody against TNFalpha used to treat Crohns, UC, RA, ankylosing spondylitis
Chlorpromazine, haloperidol Typical antipsychotics (2)
Risperidone, Clozapine, Olanzapine, Quetiapine, Ziprasidone Atypical antipsychotics (5)
Aripiprazole Antipsychotics; Dopamine system stabilizer; Partial agonist at D2 and 5-HT1a; antagonist at 5-HT2a
l-dopa, carbidopa, simemet Standard Parkinson's treatments (3)
Selegiline, Rasagiline Parkinson's treatment; MOA-B inhibitors (2)
Tolcapone, entacapone Parkinson's treatment, COMT inhibitors (prevent L-dopa breakdown in peripheral tissues) (2)
Bromocriptine, pergolide, ropinirole, pramipexole Parkinson's treatment, Dopamine agonists (4)
Benztropine, trihexyphenidyl Parkinson's treatment, centrally acting antimuscarinic agents (block muscarinics within the striatum) (2)
Amantadine Parkinson's treatment; dopamine releasing agent
Donepezil, rivastigmine, galantamine, tacrine Alzheimer's treatment; acetylcholinesterase inhibitors (4)
Memantine Alzheimer's treatment; NMDA receptor agonist
zaleplon (sonata) Hypnotic that decreases latency to sleep (~4 hr duration of action) and is approved for short term use, but has not anxiolytic or muscle relaxant properties
carbamazepine, felbamate, valproic acid Antiseizure drugs; Liver function test required by the FDA (3)
Modafinil Non-amphetamine stimulant clinically used to treat Narcolepsy
Venlafaxine, Duloxetine Antidepressants; block norephinephrine uptake as well as serotonin uptake
Sildenafil Autocoids; Prostaglandins; Trade name Viagra
Cimetidine, Ranitidine GI drugs; H2-receptor antagonist (2)
Omeprazole, Esomeprazole, Rabeprazole GI drugs; Proton pump inhibitors (3)
Diphenoxylate, loperamide, bismuth subsalicylate, alosetron GI drugs; Antidiarrheal (4)
Tegaserod, Lubiprostone GI drugs; Laxatives and stool softeners (2)
Bran, Psyllium preparations, methylcellulose GI drugs; Bulk Laxatives (3)
Milk of magnesia, sodium phosphate, glycerin, lactulose, polyethylene glycol, ascorbic acid GI drugs; Osmotically active agents (6)
Bisacodyl, cascara sagrada, senna, castor oil GI drugs; Stimulant laxatives (4)
phenobarbital, pentobarbital, thiopental Sedative-hypnotics; Barbiturates (3)
Chlordiazepoxide, diazepam, flurazepam Sedative-hypnotics, Benzodiazepines, long half-life (3)
Lorazepam, temazepam, alprazolam Sedative-hypnotics; Benzodiazepines; medium half-life (3)
Midazolam Sedative-hypnotics; Benzodiazepine; short half life
Flunitrazepam, clonazepam Sedative-hypnotics; Benzodiazepines; other (2)
Zaleplon, Zolpidem, Eszopiclone Sedative-hypnotics; Non-benzodiazepines (z-drugs); bind to BZ1 subtype of benzodiazepine sites (3)
Flumazenil Sedative-hypnotics; Non-benzodiazepines (z-drugs); benzodiazepam site antagonist
Chloral hydrate, meprobamate Sedative-hypnotics; Older sedative-hypnotics
Melatonin, Ramelteon Sedative-Hypnotics; Melatonin receptor agonists
Buspirone Sedative-hypnotic; Serotonergic agent; agonist at 5-HT1a
Diphenhydramine, doxylamine Sedative-hypnotics; Over-the-counter sleep aids; Antihistamines
Baclofen, Tizanidine, Dantrolene Sedative-hypnotics; Spasmolytics
Baclofen Sedative-hypnotics; Spasmolytic; GABAb receptor agonist
Tizanidine Sedative-hypnotics; Spasmolytic; central alpha2 receptor agonist
Hydromorphone, methadone, meperidine, fentanyl, oxycodone, loperamide, naloxone, naltrexone, buprenorphine, dextromethorphan Synthetic opiates (10)
Hydromorphone Synthetic opiate; more potent than morphine
Meperidine Synthetic opiate; less potent and shorter duration than morphine
Loperamide Synthetic opiate; controls diarrhea
Buprenorphine Synthetic opiate; partial agonist at opiate receptors, antagonizes morphine and heroin
Dextromethorphan Synthetic opiate; cough suppressant
Methotrexate, Gold, leflunomide, etanercept, infliximab, abatacept, rituximab, anakinra Inflammation; Disease-modifying anti-rheumatic drugs (8)
NSAIDs Aspirin, ibuprofen, naproxen, salicylate, celecoxib
Acetaminophen, Glucocorticoids Inflammation; others (2)
Indomethacin, colchicine, phenylbutazone Gout; Anti-inflammatory (3)
Allopurinol, febuxostat Gout; Decreased production (inhibit xanthine oxidase) (2)
Probenecid, sulfinpyrazone Gout; Uricosuric drugs
Daclizumab, basiliximab, muromonab, abatacept Immunomodulators; monoclonal antibodies used to treat inflammatory disorders (4)
cocaine, amphetamines, phenethylamine, phenylpropanolamine, kathionine Stimulants; CNS sympathomimetics (5)
methylphenidate, atomoxetine Stimulants; ADHD treatments (2)
Modafinil, gamma hydroxybutyrate Stimulants; Narcolepsy treatments (2)
Dronabinol, Rimonabant Similar to marijuana (2)
Fomepizole, Disulfiram, Naltrexone, Acamprosate Alcohol treatments (4)
Propranolol, Methysergide, Amitriptyline, verapamil, valproic acid, topiramate, gabapentin, ibuprofen Prophylactic treatments for migraine (8)
PPI/H2Ra, metronidazole, tetracycline, bismuth subsalicylate GI drugs, Antimicrobial agents, Quadruple drug therapy

Set Information

Terms 106
Creator mjswenson84
Created February 22, 2007
Groups None
Tags pharmacology, test
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mjswenson84 : Changed Antidepressants; block norephinephrine uptake as well as serotonin uptake → Venlafaxine, Duoxetine to Venlafaxine, Duloxetine → Antidepressants; block norephinephrine uptake as well as serotonin uptake
mjswenson84 : Changed Immunomodulators; monoclonal antibodies used to treat inflammatory disorders (8) → Daclizumab, basiliximab, muromonab, infliximab, etanercept, natalizumab, efalizumab, abatacept to Daclizumab, basiliximab, muromonab, abatacept → Immunomodulators; monoclonal antibodies used to treat inflammatory disorders (4)
mjswenson84 : Changed GI drugs; Antiemetics; H1 antihistamine → Dimenhydrate to GI drugs; Antiemetics; H1 antihistamine → Dimenhydrinate
mjswenson84 : Changed Gout; Anti-inflammatory (3) → Indomethacin, colchicine, phenybutazone to Indomethacin, colchicine, phenylbutazone → Gout; Anti-inflammatory (3)
mjswenson84 : Changed Indomethacin, colchicine, phenylbutazone → Gout; Anti-inflammatory (3) to Gout; Anti-inflammatory (3) → Indomethacin, colchicine, phenylbutazone
mjswenson84 : Changed Venlafaxine, Duloxetine → Antidepressants; block norephinephrine uptake as well as serotonin uptake to Antidepressants; block norephinephrine uptake as well as serotonin uptake → Venlafaxine, Duloxetine
mjswenson84 : Changed Anakinra → Immunomodulators; Cytokines and growth factors; Cytokine antagonists; IL-1 receptor antagonist to Immunomodulators; Cytokines and growth factors; Cytokine antagonists; IL-1 receptor antagonist → Anakinra
mjswenson84 : Changed Sedative-hypnotics; Benzodiazepines; medium half-life (3) → Lorazepam, temazepan, alprazolam to Sedative-hypnotics; Benzodiazepines; medium half-life (3) → Lorazepam, temazepam, alprazolam
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Most Missed Words

  1. Odansetron, granisetron, palonsetronGI drugs; Antiemetics; 5-HT3 receptor antagonists (3) - 4 misses
  2. MemantineAlzheimer's treatment; NMDA receptor agonist - 4 misses
  3. Tranylcypromine, Phenelzine, IsocarboxazidAntidepressants; MAOIs (nonselective)--Atypical depression (3) - 3 misses
  4. Lithium, Valproic acid, Carbamazepine, LamotrigineAntidepressants; For bipolar patients (4) - 3 misses
  5. Valproic acid, Lamotrigine, Topiramate, ZonisamideAntiepileptics; For a variety of seizure types (4) - 3 misses
  6. Zileuton, zafirlukast, montelukastAsthma; Anti-inflammatory agents; Leukotriene pathway modifiers (3) - 3 misses
  7. Dimenhydrinate, diphenhydramine, meclizine, promethazine, fexofenadine, loratadineAutocoids; Antihistamines (6) - 3 misses